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Pineschi M, Bertolini F, Crotti P, et al. Facile regio- and stereoselective carbon-carbon coupling of phenol derivatives with aryl aziridines. Org Lett. 2006;8(12):2627-30doi: 10.1021/ol060822m.
Pineschi, M., Bertolini, F., Crotti, P., & Macchia, F. (2006). Facile regio- and stereoselective carbon-carbon coupling of phenol derivatives with aryl aziridines. Organic letters, 8(12), 2627-30. https://doi.org/10.1021/ol060822m
Pineschi, Mauro, et al. "Facile regio- and stereoselective carbon-carbon coupling of phenol derivatives with aryl aziridines." Organic letters vol. 8,12 (2006): 2627-30. doi: https://doi.org/10.1021/ol060822m
Pineschi M, Bertolini F, Crotti P, Macchia F. Facile regio- and stereoselective carbon-carbon coupling of phenol derivatives with aryl aziridines. Org Lett. 2006 Jun 08;8(12):2627-30. doi: 10.1021/ol060822m. PMID: 16737330.
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Org Lett. 2006 Jun 08;8(12):2627-30. doi: 10.1021/ol060822m.

Facile regio- and stereoselective carbon-carbon coupling of phenol derivatives with aryl aziridines.

Organic letters

Mauro Pineschi, Ferruccio Bertolini, Paolo Crotti, Franco Macchia

Affiliations

  1. Dipartimento di Chimica Bioorganica e Biofarmacia, Università di Pisa, Via Bonanno 33, 56126 Pisa, Italy. [email protected]

PMID: 16737330 DOI: 10.1021/ol060822m

Abstract

A chemo-, regio-, and stereoselective direct carbon-carbon coupling of readily available aryl borates with N-protected aryl aziridines provides a method for the synthesis of new 2-(o-hydroxyaryl)-2-aryl ethylamines which can be used, in a novel annulation sequence, to give stereodefined substituted 3-aryl indolines. [reaction: see text]

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