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Wippich J, Schnapperelle I, Bach T. Regioselective oxidative Pd-catalysed coupling of alkylboronic acids with pyridin-2-yl-substituted heterocycles. Chem Commun (Camb). 2015;51(15):3166-8doi: 10.1039/c4cc10144h.
Wippich, J., Schnapperelle, I., & Bach, T. (2015). Regioselective oxidative Pd-catalysed coupling of alkylboronic acids with pyridin-2-yl-substituted heterocycles. Chemical communications (Cambridge, England), 51(15), 3166-8. https://doi.org/10.1039/c4cc10144h
Wippich, Julian, et al. "Regioselective oxidative Pd-catalysed coupling of alkylboronic acids with pyridin-2-yl-substituted heterocycles." Chemical communications (Cambridge, England) vol. 51,15 (2015): 3166-8. doi: https://doi.org/10.1039/c4cc10144h
Wippich J, Schnapperelle I, Bach T. Regioselective oxidative Pd-catalysed coupling of alkylboronic acids with pyridin-2-yl-substituted heterocycles. Chem Commun (Camb). 2015 Feb 21;51(15):3166-8. doi: 10.1039/c4cc10144h. PMID: 25605647.
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Chem Commun (Camb). 2015 Feb 21;51(15):3166-8. doi: 10.1039/c4cc10144h.

Regioselective oxidative Pd-catalysed coupling of alkylboronic acids with pyridin-2-yl-substituted heterocycles.

Chemical communications (Cambridge, England)

Julian Wippich, Ingo Schnapperelle, Thorsten Bach

Affiliations

  1. Department Chemie and Catalysis Research Center (CRC), Technische Universität München, 85747 Garching, Germany. [email protected].

PMID: 25605647 DOI: 10.1039/c4cc10144h

Abstract

A total of 19 alkylated heterocycles (thiophenes, benzothiophenes, pyrroles, furans) were prepared (36-99% yield) from the respective pyridin-2-yl-substituted precursors employing alkylboronic acids as the C-H alkylating reagents in an oxidative (Ag2CO3 and 2,6-dimethyl-1,4-benzoquinone as oxidants) Pd-catalysed coupling reaction.

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