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Kimura O, Fujii Y, Haraguchi K, et al. Effects of perfluoroalkyl carboxylic acids on the uptake of sulfobromophthalein via organic anion transporting polypeptides in human intestinal Caco-2 cells. Biochem Biophys Rep. 2020;24:100807doi: 10.1016/j.bbrep.2020.100807.
Kimura, O., Fujii, Y., Haraguchi, K., Kato, Y., Ohta, C., Koga, N., & Endo, T. (2020). Effects of perfluoroalkyl carboxylic acids on the uptake of sulfobromophthalein via organic anion transporting polypeptides in human intestinal Caco-2 cells. Biochemistry and biophysics reports, 24100807. https://doi.org/10.1016/j.bbrep.2020.100807
Kimura, Osamu, et al. "Effects of perfluoroalkyl carboxylic acids on the uptake of sulfobromophthalein via organic anion transporting polypeptides in human intestinal Caco-2 cells." Biochemistry and biophysics reports vol. 24 (2020): 100807. doi: https://doi.org/10.1016/j.bbrep.2020.100807
Kimura O, Fujii Y, Haraguchi K, Kato Y, Ohta C, Koga N, Endo T. Effects of perfluoroalkyl carboxylic acids on the uptake of sulfobromophthalein via organic anion transporting polypeptides in human intestinal Caco-2 cells. Biochem Biophys Rep. 2020 Sep 07;24:100807. doi: 10.1016/j.bbrep.2020.100807. eCollection 2020 Dec. PMID: 32964147; PMCID: PMC7490525.
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Biochem Biophys Rep. 2020 Sep 07;24:100807. doi: 10.1016/j.bbrep.2020.100807. eCollection 2020 Dec.

Effects of perfluoroalkyl carboxylic acids on the uptake of sulfobromophthalein via organic anion transporting polypeptides in human intestinal Caco-2 cells.

Biochemistry and biophysics reports

Osamu Kimura, Yukiko Fujii, Koichi Haraguchi, Yoshihisa Kato, Chiho Ohta, Nobuyuki Koga, Tetsuya Endo

Affiliations

  1. School of Pharmaceutical Sciences, Health Sciences University of Hokkaido, 1757 Kanazawa, Ishikari-Tobetsu, Hokkaido, 061-0293, Japan.
  2. Daiichi University of Pharmacy, Tamagawa-cho, Minami-ku, Fukuoka, 815-8511, Japan.
  3. Kagawa School of Pharmaceutical Sciences, Tokushima Bunri University, Sanuki, Kagawa, 769-2193, Japan.
  4. Faculty of Nutritional Sciences, Nakamura Gakuen University, Johnan-ku, Fukuoka, 814-0198, Japan.

PMID: 32964147 PMCID: PMC7490525 DOI: 10.1016/j.bbrep.2020.100807

Abstract

We performed a detailed investigation of the uptake of sulfobromophthalein (BSP) from the apical membrane of Caco-2 cells, which is a substrate for organic anion transporting polypeptides (OATPs), and calculated the kinetic parameters of BSP uptake as follows: K

© 2020 The Authors.

Keywords: Caco-2 cells; Intestinal absorption; Organic anion transport polypeptides (OATPs); Perfluoroalkyl carboxylic acids (PFCAs); Sulfobromophthalein (BSP)

Conflict of interest statement

The authors declare that there are no conflicts of interest.

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