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Purinergic Signal. 2021 Sep;17(3):503-514. doi: 10.1007/s11302-021-09806-6. Epub 2021 Jul 27.

Lack of efficacy of a partial adenosine A1 receptor agonist in neuropathic pain models in mice.

Purinergic signalling

Katharina Metzner, Tilman Gross, Annika Balzulat, Gesine Wack, Ruirui Lu, Achim Schmidtko

Affiliations

  1. Institute of Pharmacology and Clinical Pharmacy, Goethe University Frankfurt, 60438, Frankfurt am Main, Germany. [email protected].
  2. Institute of Pharmacology and Clinical Pharmacy, Goethe University Frankfurt, 60438, Frankfurt am Main, Germany.

PMID: 34313915 PMCID: PMC8410902 DOI: 10.1007/s11302-021-09806-6

Abstract

Previous studies suggest that adenosine A

© 2021. The Author(s).

Keywords: Adenosine A1 receptor; In situ hybridization; Neuropathic pain; Pain behavior; Partial agonist; Patch-clamp

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