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Xenobiotica. 2021 Nov 07;1-12. doi: 10.1080/00498254.2021.2002973. Epub 2021 Nov 07.

The Metabolism and Excretion of the Dipeptidyl Peptidase 4 Inhibitor [.

Xenobiotica; the fate of foreign compounds in biological systems

Jinmiao Lu, Yicong Bian, Hua Zhang, Dong Tang, Xusheng Tian, Xinyi Zhou, Zengyan Xu, Yating Xiong, Zheming Gu, Zhenwen Yu, Tong Wang, Juping Ding, Qiang Yu, Jinsong Ding

Affiliations

  1. Xiangya School of Pharmaceutical Sciences, Central South University, Hunan, China.
  2. CGeneTech (Suzhou, China) Co., Ltd, Jiangsu, China.
  3. Department of Clinical Pharmacology, the First Affiliated Hospital of Soochow University, Suzhou, China.
  4. Value Pharmaceutical Services Co., Ltd, Jiangsu, China.

PMID: 34743655 DOI: 10.1080/00498254.2021.2002973

Abstract

1. The metabolism and excretion of cetagliptin were investigated in healthy male subjects after a single oral dose of 100mg/50μCi [

Keywords: cetagliptin; excretion; healthy subjects; metabolism; metabolite

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