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Vachal P, Duffy JL, Campeau LC, et al. Invention of MK-8262, a Cholesteryl Ester Transfer Protein (CETP) Inhibitor Backup to Anacetrapib with Best-in-Class Properties. J Med Chem. 2021;64(18):13215-13258doi: 10.1021/acs.jmedchem.1c00959.
Vachal, P., Duffy, J. L., Campeau, L. C., Amin, R. P., Mitra, K., Murphy, B. A., Shao, P. P., Sinclair, P. J., Ye, F., Katipally, R., Lu, Z., Ondeyka, D., Chen, Y. H., Zhao, K., Sun, W., Tyagarajan, S., Bao, J., Wang, S. P., Cote, J., Lipardi, C., Metzger, D., Leung, D., Hartmann, G., Wollenberg, G. K., Liu, J., Tan, L., Xu, Y., Chen, Q., Liu, G., Blaustein, R. O., & Johns, D. G. (2021). Invention of MK-8262, a Cholesteryl Ester Transfer Protein (CETP) Inhibitor Backup to Anacetrapib with Best-in-Class Properties. Journal of medicinal chemistry, 64(18), 13215-13258. https://doi.org/10.1021/acs.jmedchem.1c00959
Vachal, Petr, et al. "Invention of MK-8262, a Cholesteryl Ester Transfer Protein (CETP) Inhibitor Backup to Anacetrapib with Best-in-Class Properties." Journal of medicinal chemistry vol. 64,18 (2021): 13215-13258. doi: https://doi.org/10.1021/acs.jmedchem.1c00959
Vachal P, Duffy JL, Campeau LC, Amin RP, Mitra K, Murphy BA, Shao PP, Sinclair PJ, Ye F, Katipally R, Lu Z, Ondeyka D, Chen YH, Zhao K, Sun W, Tyagarajan S, Bao J, Wang SP, Cote J, Lipardi C, Metzger D, Leung D, Hartmann G, Wollenberg GK, Liu J, Tan L, Xu Y, Chen Q, Liu G, Blaustein RO, Johns DG. Invention of MK-8262, a Cholesteryl Ester Transfer Protein (CETP) Inhibitor Backup to Anacetrapib with Best-in-Class Properties. J Med Chem. 2021 Sep 23;64(18):13215-13258. doi: 10.1021/acs.jmedchem.1c00959. Epub 2021 Aug 10. PMID: 34375108.
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