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Come JH, Senter TJ, Clark MP, et al. Discovery and Optimization of Pyrazole Amides as Inhibitors of ELOVL1. J Med Chem. 2021;64(24):17753-17776doi: 10.1021/acs.jmedchem.1c00944.
Come, J. H., Senter, T. J., Clark, M. P., Court, J. J., Gale-Day, Z., Gu, W., Krueger, E., Liang, J., Morris, M., Nanthakumar, S., O'Dowd, H., Maltais, F., Iyer, G., Andreassi, J., Boucher, C., Considine, T., Moody, C. S., Taylor, W., Mohanty, A. K., Huang, Y., Zuccola, H., Coll, J., Bonanno, K. C., Gagnon, K. J., Gan, L., Lu, F., Gao, H., Chakilam, A., Engtrakul, J., Song, B., Crawford, D., Doyle, E., Kramer, T., Vought, B., Phillips, J., Kemper, R., Sanders, M., Swett, R., Furey, B., Winquist, R., Bunnage, M. E., Jackson, K. L., Charifson, P. S., & Magavi, S. S. (2021). Discovery and Optimization of Pyrazole Amides as Inhibitors of ELOVL1. Journal of medicinal chemistry, 64(24), 17753-17776. https://doi.org/10.1021/acs.jmedchem.1c00944
Come, Jon H, et al. "Discovery and Optimization of Pyrazole Amides as Inhibitors of ELOVL1." Journal of medicinal chemistry vol. 64,24 (2021): 17753-17776. doi: https://doi.org/10.1021/acs.jmedchem.1c00944
Come JH, Senter TJ, Clark MP, Court JJ, Gale-Day Z, Gu W, Krueger E, Liang J, Morris M, Nanthakumar S, O'Dowd H, Maltais F, Iyer G, Andreassi J, Boucher C, Considine T, Moody CS, Taylor W, Mohanty AK, Huang Y, Zuccola H, Coll J, Bonanno KC, Gagnon KJ, Gan L, Lu F, Gao H, Chakilam A, Engtrakul J, Song B, Crawford D, Doyle E, Kramer T, Vought B, Phillips J, Kemper R, Sanders M, Swett R, Furey B, Winquist R, Bunnage ME, Jackson KL, Charifson PS, Magavi SS. Discovery and Optimization of Pyrazole Amides as Inhibitors of ELOVL1. J Med Chem. 2021 Dec 23;64(24):17753-17776. doi: 10.1021/acs.jmedchem.1c00944. Epub 2021 Nov 08. PMID: 34748351.
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