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ChemistryOpen. 2019 Jun 07;8(6):737-742. doi: 10.1002/open.201900110. eCollection 2019 Jun.

Conjugates of Cryptophycin and RGD or .

ChemistryOpen

Adina Borbély, Eduard Figueras, Ana Martins, Lizeth Bodero, André Raposo Moreira Dias, Paula López Rivas, Arianna Pina, Daniela Arosio, Paola Gallinari, Marcel Frese, Christian Steinkühler, Cesare Gennari, Umberto Piarulli, Norbert Sewald

Affiliations

  1. Organic and Bioorganic Chemistry, Department of Chemistry Bielefeld University Universitätsstraße 25 DE-33615 Bielefeld Germany.
  2. Exiris s.r.l. Via di Castel Romano 100 IT-00128 Rome Italy.
  3. Dipartimento di Scienza e Alta Tecnologia Università degli Studi dell'Insubria Via Valleggio, 11 IT-22100 Como Italy.
  4. Dipartimento di Chimica Università degli Studi di Milano Via C. Golgi, 19 IT-20133 Milano Italy.
  5. Istituto di Scienze e Tecnologie Molecolari (ISTM) CNR Via C. Golgi, 19 IT-20133 Milano Italy.

PMID: 31275795 PMCID: PMC6587324 DOI: 10.1002/open.201900110

Abstract

RGD-cryptophycin and

Keywords: antitumor agents; cancer; drug delivery; integrins; peptidomimetics

Conflict of interest statement

A.M. is an employee of Exiris, P.G. is a shareholder of Exiris. C.S. is a shareholder of Exiris.

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