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Machulkin AE, Uspenskaya AA, Zyk NU, et al. Synthesis, Characterization, and Preclinical Evaluation of a Small-Molecule Prostate-Specific Membrane Antigen-Targeted Monomethyl Auristatin E Conjugate. J Med Chem. 2021;64(23):17123-17145doi: 10.1021/acs.jmedchem.1c01157.
Machulkin, A. E., Uspenskaya, A. A., Zyk, N. U., Nimenko, E. A., Ber, A. P., Petrov, S. A., Polshakov, V. I., Shafikov, R. R., Skvortsov, D. A., Plotnikova, E. A., Pankratov, A. A., Smirnova, G. B., Borisova, Y. A., Pokrovsky, V. S., Kolmogorov, V. S., Vaneev, A. N., Khudyakov, A. D., Chepikova, O. E., Kovalev, S., Zamyatnin, A. A., Erofeev, A., Gorelkin, P., Beloglazkina, E. K., Zyk, N. V., Khazanova, E. S., & Majouga, A. G. (2021). Synthesis, Characterization, and Preclinical Evaluation of a Small-Molecule Prostate-Specific Membrane Antigen-Targeted Monomethyl Auristatin E Conjugate. Journal of medicinal chemistry, 64(23), 17123-17145. https://doi.org/10.1021/acs.jmedchem.1c01157
Machulkin, Aleksei E, et al. "Synthesis, Characterization, and Preclinical Evaluation of a Small-Molecule Prostate-Specific Membrane Antigen-Targeted Monomethyl Auristatin E Conjugate." Journal of medicinal chemistry vol. 64,23 (2021): 17123-17145. doi: https://doi.org/10.1021/acs.jmedchem.1c01157
Machulkin AE, Uspenskaya AA, Zyk NU, Nimenko EA, Ber AP, Petrov SA, Polshakov VI, Shafikov RR, Skvortsov DA, Plotnikova EA, Pankratov AA, Smirnova GB, Borisova YA, Pokrovsky VS, Kolmogorov VS, Vaneev AN, Khudyakov AD, Chepikova OE, Kovalev S, Zamyatnin AA, Erofeev A, Gorelkin P, Beloglazkina EK, Zyk NV, Khazanova ES, Majouga AG. Synthesis, Characterization, and Preclinical Evaluation of a Small-Molecule Prostate-Specific Membrane Antigen-Targeted Monomethyl Auristatin E Conjugate. J Med Chem. 2021 Dec 09;64(23):17123-17145. doi: 10.1021/acs.jmedchem.1c01157. Epub 2021 Nov 19. PMID: 34797052.
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